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Compile Data Set for Download or QSAR
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Found
1
Enz. Inhib. hit(s) with Target = 'Estrogen receptor [Y537S]' and Ligand = 'BDBM263716'
Target
Estrogen receptor [Y537S]
(Homo sapiens (Human))
Sanofi
US Patent
Ligand
BDBM263716
(6-(2,4-dichlorophenyl)-5-[4-[(3S)-1-(3-fluoropropy...)
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Affinity Data
IC50: 221nM
pH: 7.4 T: 2°C
Assay Description:
It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...
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Target Info
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Ligand Info
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3D Structure (crystal)
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