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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor beta' and Ligand = 'BDBM50551582'
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50551582(CHEMBL279301 | E-4-Hydroxytamoxifen)
Affinity DataIC50:  0.990nMAssay Description:Antagonist activity at ERbeta (unknown origin) expressed in human U2OS cells assessed as inhibition of E2-induced transactivation measured after 21 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50551582(CHEMBL279301 | E-4-Hydroxytamoxifen)
Affinity DataIC50:  1.70nMAssay Description:Displacement of fluorescent-labelled E2 from recombinant human GST-tagged ERbeta by LanthaScreen TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed