Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Extracellular calcium-sensing receptor' and Ligand = 'BDBM50133679'
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  3.47E+5nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50133679(CHEMBL3633665)
Affinity DataIC50:  3.47E+5nMAssay Description:Antagonist activity at rat CaSR expressed in HEK293 cells assessed as inhibition of Ca2+-induced inositol monophosphate accumulation after 1 hr by FR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed