Report error Found 7 Enz. Inhib. hit(s) with Target = 'Focal adhesion kinase 1' and Ligand = 'BDBM50246060'
Affinity DataIC50: 1nMAssay Description:Inhibition of purified activated FAK kinase domain (410-689) using ATP and Glu and Tyr random peptide polymer substrate by fluorescence polarization ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of GST-tagged FAK assessed as inhibition of poly-Glu-Tyr phosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of purified-activated FAK kinase domain (amino acids 410-689) (unknown origin) using Glu and Tyr, p(Glu/Tyr) peptide in presence of ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of full-length C-terminal his-tagged human FAK pre-incubated with enzyme for 1 h prior to the addition of 500 uM ATPMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Inhibition of full-length FAK (unknown origin) with N-terminal NanoLuc-fusion expressed in HEK293T cells by NanoBRET assayMore data for this Ligand-Target Pair
