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Found 6 Enz. Inhib. hit(s) with Target = 'Free fatty acid receptor 1' and Ligand = 'BDBM50275597'
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275597(3-(4-(o-Tolylethynyl)phenyl)propanoic acid | CHEMB...)
Affinity DataKi:  631nMAssay Description:Displacement of 3-(2-Fluoro-4-((2'-methyl-4'-(2-(2-((7-nitrobenzo[c][1,2,5]-oxadiazol-4-yl)amino)ethoxy)ethoxy)-[1,1'-biphenyl]-3-yl)-methoxy)phenyl)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275597(3-(4-(o-Tolylethynyl)phenyl)propanoic acid | CHEMB...)
Affinity DataEC50:  45.7nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells assessed as calcium mobilization by fluorescence spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275597(3-(4-(o-Tolylethynyl)phenyl)propanoic acid | CHEMB...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human FFA1 receptor transfected in human 1321N1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275597(3-(4-(o-Tolylethynyl)phenyl)propanoic acid | CHEMB...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human FFA1 assessed as calcium mobilization measured for 50 intervals of 0.4 secs by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275597(3-(4-(o-Tolylethynyl)phenyl)propanoic acid | CHEMB...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at human FFA1 expressed in human 1321N1 cells by calcium fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark

Curated by ChEMBL
LigandPNGBDBM50275597(3-(4-(o-Tolylethynyl)phenyl)propanoic acid | CHEMB...)
Affinity DataEC50:  68nMAssay Description:Agonist activity at human C-terminal eYFP-tagged FFA1 receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment incubated for 5 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed