Affinity DataIC50: 700nMAssay Description:Inhibition of recombinant HA-tagged K-Ras G12V mutant (unknown origin) assessed as disruption of interaction with GST-tagged Raf-RBD after overnight ...More data for this Ligand-Target Pair
Affinity DataKd: 830nMAssay Description:Binding affinity to K-Ras G12V mutant (unknown origin) after 2 hrs by fluorescence polarization-based spectrofluorimetric analysisMore data for this Ligand-Target Pair