Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'GTPase KRas' and Ligand = 'BDBM50549223'
TargetGTPase KRas(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50549223(CHEMBL4796065)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of C-terminal Avi-tagged biotinylated KRas G12D mutant (1 to 169 residues) (unknown origin) expressed in Escherichia coli assessed as redu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGTPase KRas(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50549223(CHEMBL4796065)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to GCP-KRAS G12D (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB