Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'GTPase KRas' and Ligand = 'BDBM50585384'
TargetGTPase KRas(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50585384(CHEMBL5084171)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to wild type KRAS (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetGTPase KRas(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50585384(CHEMBL5084171)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to human AviTEV6His-tagged KRAS isoform 4B wild type (1 to 169 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissoc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB