Found 3 Enz. Inhib. hit(s) with Target = 'Gastrin/cholecystokinin type B receptor' and Ligand = 'BDBM50549227' TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Medical University Of Innsbruck
Curated by ChEMBL
Medical University Of Innsbruck
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I][3-iodo Tyr12,Leu15]gastrin-I from human CCK2R expressed in human A431 cells measured after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Medical University Of Innsbruck
Curated by ChEMBL
Medical University Of Innsbruck
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at human CCK2R expressed in human A431 cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye ba...More data for this Ligand-Target Pair
