Affinity DataIC50: 21nMAssay Description:Antagonist activity against human glucagon receptor expressed in CHO cell membranes using [125I]glucagonMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity to GlucR in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Binding affinity to human cloned GluR expressed in BHK cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 144nMAssay Description:Inhibitory concentration against glucagon-induced cAMP accumulation in human glucagon receptor transfected CHO cellsMore data for this Ligand-Target Pair