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Found 3 Enz. Inhib. hit(s) with Target = 'Glutamate receptor 1' and Ligand = 'BDBM50166285'
TargetGlutamate receptor 1(Rattus norvegicus (Rat))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50166285((RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazo...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]AMPA from rat recombinant GluR1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50166285((RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazo...)
Affinity DataKi:  5.15E+3nMAssay Description:Binding affinity for ionotropic Glutamate receptor AMPA 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 1(Homo sapiens (Human))
The Danish University Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50166285((RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazo...)
Affinity DataEC50:  4.80E+5nMAssay Description:Agonist activity at GluR1 expressed in HEK293 cells by Fluo-4/Ca2+ assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed