Found 3 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 2' and Ligand = 'BDBM50088213'
Affinity DataKi: 1.84E+3nMAssay Description:compound was tested for binding affinity against human Ionotropic glutamate receptor ionotropic kainate 2 in HK293 cells using [3H]-kainate as radiol...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+4nMAssay Description:Agonist activity at iGluR6 L439C mutant expressed in human HEK293 cells assessed as increase in intracellular Ca2+ levels by FURA-2-M staining based ...More data for this Ligand-Target Pair
Affinity DataEC50: 8.30E+3nMAssay Description:Effective concentration against human GluR6 expressed in HEK293 cellsMore data for this Ligand-Target Pair