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Found 2 Enz. Inhib. hit(s) with Target = 'Glutaminase kidney isoform, mitochondrial' and Ligand = 'BDBM332753'
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM332753((2S)-2-[3-(Trifluoromethoxy)phenyl]-2-methoxy-N-[6...)
Affinity DataIC50:  95.7nMAssay Description:A Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity of GLS1 in vitro. 6His t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Cancer Research Technology

US Patent
LigandPNGBDBM332753((2S)-2-[3-(Trifluoromethoxy)phenyl]-2-methoxy-N-[6...)
Affinity DataIC50:  95.7nMAssay Description:GLS Enzyme Potency AssayA Glutamate Oxidase/AmplexRed coupled assay was used to measure the ability of compounds to bind to and inhibit the activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent