Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Glutaminyl-peptide cyclotransferase' and Ligand = 'BDBM50439173'
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50439173(CHEMBL2418770)
Affinity DataKi:  1.14E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Escherichia coli DH5alpha using H-Gln-AMC as substrate by fluorometric analysis in presence of py...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug

Curated by ChEMBL
LigandPNGBDBM50439173(CHEMBL2418770)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of human glutaminyl cyclase expressed in Escherichia coli DH5alpha using H-Gln-AMC as substrate by fluorometric analysis in presence of py...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed