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Found 2 Enz. Inhib. hit(s) with Target = 'High affinity choline transporter 1' and Ligand = 'BDBM50067201'
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50067201(CHEMBL3186365)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells assessed as remaining transporter activity in presence of 10 uM [3H]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50067201(CHEMBL3186365)
Affinity DataIC50:  8.09E+3nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells assessed as remaining transporter activity in presence of 100 nM [3H...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed