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Found 2 Enz. Inhib. hit(s) with Target = 'High affinity choline transporter 1' and Ligand = 'BDBM87569'
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM87569(MLS000733239 | N-(1-phenylethyl)-4-[1-(pyridin-2-y...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells by membrane depolarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM87569(MLS000733239 | N-(1-phenylethyl)-4-[1-(pyridin-2-y...)
Affinity DataIC50:  1.79E+3nMAssay Description:Data Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center Affiliation: Johns Hopkins University, School of Medicine Screening ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay