Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'High affinity choline transporter 1' and Ligand = 'BDBM87575'
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay
LigandPNGBDBM87575(MLS001126544 | N-[(4,5-dimethyl-1,3-thiazol-2-yl)m...)
Affinity DataIC50:  303nMAssay Description:Data Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center Affiliation: Johns Hopkins University, School of Medicine Screening ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Johns Hopkins Ion Channel Center

Curated by PubChem BioAssay
LigandPNGBDBM87575(MLS001126544 | N-[(4,5-dimethyl-1,3-thiazol-2-yl)m...)
Affinity DataIC50:  760nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells by membrane depolarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed