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Found 2 Enz. Inhib. hit(s) with Target = 'High affinity choline transporter 1' and Ligand = 'BDBM87577'
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM87577(3-[(1-isopropyl-4-piperidyl)oxy]-4-methoxy-N-(1-me...)
Affinity DataIC50:  4.47E+3nMAssay Description:Inhibition of human CHT Leu530Ala and Val531Ala mutant expressed in HEK293 cells by membrane depolarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity choline transporter 1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM87577(3-[(1-isopropyl-4-piperidyl)oxy]-4-methoxy-N-(1-me...)
Affinity DataIC50:  7.51E+3nMAssay Description:Data Source (MLPCN Center Name): Johns Hopkins Ion Channel Center (JHICC) Center Affiliation: Johns Hopkins University, School of Medicine Screening ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay