Found 11 Enz. Inhib. hit(s) with Target = 'Histamine H1 receptor' and Ligand = 'BDBM50017674' TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKi: 14.8nMAssay Description:Displacement of [3H]mepyramine from human H1R expressed in Sf9 cells co-expressing RGS4 after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataIC50: 8.40E+4nMAssay Description:Affinities of the test compounds for peripheral human histamine H-4-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataIC50: 8.40E+4nMAssay Description:The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine...More data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
University of North Carolina At Chapel Hill
Curated by PDSP Ki Database
Affinity DataKd: 11.8nMAssay Description:Antagonist activity at H1R in guinea pig ileum assessed as inhibition of histamine-induced muscle contraction after 15 minsMore data for this Ligand-Target Pair
