TargetHistamine H3 receptor(Rattus norvegicus (rat))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from histamine H3 receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Binding affinity against H3 receptor in rat cerebral cortex membranes was evaluated using [3H]N-methyl-histamine as radioligandMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Heinrich Heine University D£Sseldorf
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair