Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.730nMAssay Description:Inverse agonist activity at human histamine H3 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair