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Found 2 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT2B' and Ligand = 'BDBM311486'
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM311486(CHEM-US-00192 | US10155764, Example 65B)
Affinity DataIC50:  19nMAssay Description:Inhibition of biotinylated ligand binding to FLAG epitope-fused/His-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) measured after 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM311486(CHEM-US-00192 | US10155764, Example 65B)
Affinity DataIC50:  19nMAssay Description:Displacement of biotinylated small molecule ligand from His/FLAG-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) after 15 mins by Alph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed