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Found 2 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT2B' and Ligand = 'BDBM50512967'
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50512967(CHEMBL4449143)
Affinity DataIC50:  14nMAssay Description:Inhibition of biotinylated peptide binding to human GST-tagged PCAF bromodomain expressed in Escherichia coli Rosetta (DE3) measured after 15 hrs by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50512967(CHEMBL4449143)
Affinity DataKd:  118nMAssay Description:Binding affinity to human N-terminal His-tagged PCAF by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed