Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase KAT2B' and Ligand = 'BDBM50512980'
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50512980(CHEMBL4570969)
Affinity DataIC50:  36nMAssay Description:Inhibition of biotinylated peptide binding to human GST-tagged PCAF bromodomain expressed in Escherichia coli Rosetta (DE3) measured after 15 hrs by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50512980(CHEMBL4570969)
Affinity DataKd:  126nMAssay Description:Binding affinity to human PCAF bromodomain by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed