Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase p300' and Ligand = 'BDBM50081125'
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50081125(CHEMBL3421961)
Affinity DataKi:  2.00E+3nMAssay Description:Noncompetitive inhibition of P300 (unknown origin) using acetyl CoA as substrate after 15 mins by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50081125(CHEMBL3421961)
Affinity DataKi:  9.40E+3nMAssay Description:Noncompetitive inhibition of P300 (unknown origin) using biotinylated H3 as substrate after 15 mins by double reciprocal plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50081125(CHEMBL3421961)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of recombinant P300 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed