Found 6 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase p300' and Ligand = 'BDBM50241990' TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataKi: 4.90E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant histone acetyltransferase p300 (unknown origin) using dH3-H4 tetramer and [3H]-acetyl-CoA assessed as acetate incorporation...More data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of HAT p300More data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataKd: 6.60E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataKd: 400nMT: 2°CAssay Description:The p300 activity assays were performed by a colorimetric kit (JM-K322-100, MBL) using active recombinant p300/HAT as positive control and acetyl-CoA...More data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by fluorometric titrationMore data for this Ligand-Target Pair
