Found 3 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase p300' and Ligand = 'BDBM50377962'
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataKi: 3.90E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by fluorometric titrationMore data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Jawaharlal Nehru Centre For Advanced Scientific Research
Curated by ChEMBL
Affinity DataKd: 5.90E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by isothermal titration calorimetryMore data for this Ligand-Target Pair