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Found 3 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase p300' and Ligand = 'BDBM50377962'
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50377962(CAMBOGIN)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of HAT p300 catalytic domain by equilibrium dialysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50377962(CAMBOGIN)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by fluorometric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Jawaharlal Nehru Centre For Advanced Scientific Research

Curated by ChEMBL
LigandPNGBDBM50377962(CAMBOGIN)
Affinity DataKd:  5.90E+3nMAssay Description:Binding affinity to HAT p300 catalytic domain by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed