Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 4 [653-1084,H976Y]' and Ligand = 'BDBM25175'
TargetHistone deacetylase 4 [653-1084,H976Y](Homo sapiens (Human))
Irbm/Merck Research Laboratories

LigandPNGBDBM25175(1-(5-{[benzyl(methyl)amino]methyl}thiophen-2-yl)-2...)
Affinity DataIC50:  1.10E+3nMT: 2°CAssay Description:The Fluor-de-Lys HDAC activity assay kit (Biomol) was used. Purified recombinant HDAC enzyme was incubated with Fluor-de-Lys substrate in the presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed