Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase NSD3' and Ligand = 'BDBM50608080'
TargetHistone-lysine N-methyltransferase NSD3(Homo sapiens (Human))TBA
LigandPNGBDBM50608080(CHEMBL5277519)
Affinity DataIC50:  203nMAssay Description:Antagonist activity against recombinant human GST-tagged NSD3 PWWP1 domain (247 to 398 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase NSD3(Homo sapiens (Human))TBA
LigandPNGBDBM50608080(CHEMBL5277519)
Affinity DataKd:  1.66E+5nMAssay Description:Binding affinity to recombinant human NSD3 PWWP1 domain (247 to 398 residues) by SPR analysisMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed