Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Homeodomain-interacting protein kinase 2' and Ligand = 'BDBM17055'
TargetHomeodomain-interacting protein kinase 2(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIPK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHomeodomain-interacting protein kinase 2(Homo sapiens (Human))
Masaryk University

Curated by ChEMBL
LigandPNGBDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)
Affinity DataKd:  140nMAssay Description:Binding constant for HIPK2 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed