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Found 5 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50184347'
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  430nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by gel-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50: >4.10E+3nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MnCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity in presence of MgCl2 by plate-based electrochemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184347((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-4-oxo-...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity in presence of MgCl2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed