Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Integrin alpha-V/beta-3' and Ligand = 'BDBM50318878'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50318878((S)-3-(3-methoxy-4-(4-(1,4,5,6-tetrahydropyrimidin...)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of integrin alphaVbeta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50318878((S)-3-(3-methoxy-4-(4-(1,4,5,6-tetrahydropyrimidin...)
Affinity DataIC50:  0.190nMAssay Description:Antagonist activity at alphavbeta3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50318878((S)-3-(3-methoxy-4-(4-(1,4,5,6-tetrahydropyrimidin...)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at alphavbeta3 integrin receptor human VSMC assessed as inhibition of vitronectin-induced cell adhesionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed