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Found 1 Enz. Inhib. hit(s) with Target = 'Interstitial collagenase' and Ligand = 'BDBM11553'
TargetInterstitial collagenase(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM11553((3R)-2-[(4-tert-butyl-1,1-biphenyl-4-yl)methyl]-N-...)
Affinity DataKi:  3.17E+3nM ΔG°:  -31.4kJ/molepH: 7.5 T: 2°CAssay Description:The enzymatic activities of MMPs were determined with recombinant human version catalytic domains and a fluorogenic peptide substrate. Fluorescence m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed