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Found 1 Enz. Inhib. hit(s) with Target = 'Kallikrein-5 [D153N]' and Ligand = 'BDBM113248'
TargetKallikrein-5 [D153N](Homo sapiens (Human))
Sixera Pharma

US Patent
LigandPNGBDBM113248(US9695194, 7)
Affinity DataKi:  2.20E+3nM ΔG°:  -33.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In DepthDetails US Patent