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Found 5 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50029783'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  491nMAssay Description:Inhibition of radioligand [3H]U69,593 binding to kappa 1 receptor of guinea pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataKi:  2.54E+3nMAssay Description:Ability to inhibit [3H]-U69,593 binding to guinea pig Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataIC50:  2.02E+3nMAssay Description:Inhibition of [3H]U-69593 radioligand binding to Guinea pig opioid receptor kappa 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataIC50:  2.03E+3nMAssay Description:Compound was evaluated for inhibition of binding of [3H]- U69,593 to Guinea pig Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50029783(5-(3-Hydroxy-phenyl)-2-methyl-2-aza-bicyclo[3.3.1]...)
Affinity DataIC50:  5.07E+3nMAssay Description:Inhibition of [3H]- U69,593 binding to Guinea pig Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed