Affinity DataKi: 470nMAssay Description:Binding affinity for 1 uM [3H]-diprenorphine against human Opioid receptor kappa expressed in chinese hamster ovary cells (CHO cells)More data for this Ligand-Target Pair
Affinity DataEC50: 227nMAssay Description:Concentration required to enhance [35S]-GTP-gammaS, binding to human Opioid receptor kappa expressed in CHO cellsMore data for this Ligand-Target Pair