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Found 2 Enz. Inhib. hit(s) with Target = 'L-lactate dehydrogenase A chain' and Ligand = 'BDBM50192453'
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50192453(AMP(2-) | Adenosine-5-monophosphate | LDHA Inhibit...)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM50192453(AMP(2-) | Adenosine-5-monophosphate | LDHA Inhibit...)
Affinity DataKd:  6.50E+5nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed