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Found 4 Enz. Inhib. hit(s) with Target = 'L-lactate dehydrogenase A chain' and Ligand = 'BDBM50425798'
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425798(CHEMBL2316886)
Affinity DataIC50:  220nMAssay Description:Inhibition of LDH-A (unknown origin) in absence of 0.1% TritonMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425798(CHEMBL2316886)
Affinity DataIC50:  325nMAssay Description:Inhibition of LDH-A (unknown origin) in presence of 0.1% TritonMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425798(CHEMBL2316886)
Affinity DataIC50:  440nMAssay Description:Inhibition of LDH-A (unknown origin) by cell based assayMore data for this Ligand-Target Pair
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425798(CHEMBL2316886)
Affinity DataKd:  68nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair