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Found 3 Enz. Inhib. hit(s) with Target = 'L-lactate dehydrogenase A chain' and Ligand = 'BDBM50433843'
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50433843(CHEMBL2382401)
Affinity DataIC50:  480nMAssay Description:Inhibition of LDHA (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50433843(CHEMBL2382401)
Affinity DataIC50:  480nMAssay Description:Inhibition of human recombinant carboxy-terminal his-tagged LDHA (1 to 331) expressed in Escherichia coli using pyruvate as substrate after 10 mins b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50433843(CHEMBL2382401)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to human recombinant carboxy-terminal avi-tagged LDHA (1 to 331) expressed in Escherichia coli by surface plasmon resonance analysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed