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Found 2 Enz. Inhib. hit(s) with Target = 'L-lactate dehydrogenase A chain' and Ligand = 'BDBM50539402'
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Jilin University China-Japan Union Hospital

Curated by ChEMBL
LigandPNGBDBM50539402(CHEMBL4645847)
Affinity DataKd:  9.85E+3nMAssay Description:Binding affinity at human LDHA assessed as dissociation constant by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
Jilin University China-Japan Union Hospital

Curated by ChEMBL
LigandPNGBDBM50539402(CHEMBL4645847)
Affinity DataEC50:  3.26E+3nMAssay Description:Inhibition of human LDHA using NADH and pyruvate by microplate reader based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed