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Found 1 Enz. Inhib. hit(s) with Target = 'MAP/microtubule affinity-regulating kinase 3' and Ligand = 'BDBM107110'
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM107110(US8592425, 14)
Affinity DataIC50:  15nMAssay Description:MARK3 activity was assayed in vitro using a Cdc25C biotinylated peptide substrate (Cell Signalling Technologies). The phosphopeptide product was quan...More data for this Ligand-Target Pair
In DepthDetails US Patent