Found 1 Enz. Inhib. hit(s) with Target = 'MAP kinase-interacting serine/threonine-protein kinase 1/2' and Ligand = 'BDBM375353'
TargetMAP kinase-interacting serine/threonine-protein kinase 1/2(Homo sapiens (Human))
Agency For Science, Technology And Research (A*Star)
Curated by ChEMBL
Agency For Science, Technology And Research (A*Star)
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of MNK1/2 in human HeLa cells assessed as decrease in eIF4E phosphorylation at Ser209 after 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair