Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit [V559D,T670I]' and Ligand = 'BDBM504400'
TargetMast/stem cell growth factor receptor Kit [V559D,T670I](Homo sapiens (Human))
Blueprint Medicines

US Patent
LigandPNGBDBM504400((S)-4-(4-(5-(1-amino-1-(4-fluorophenyl)ethyl)pyrim...)
Affinity DataIC50:  5.5nMAssay Description:KIT, KIT mutant, and PDGFRα mutant kinase profiling was performed with recombinant enzymes including wild-type KIT, KIT V560G, KIT V559D/T670I, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent