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Found 3 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM142203'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM142203(US8933079, 7.12 | US8933079, 7.13)
Affinity DataIC50:  30nMpH: 7.0Assay Description:Membranes from CHO/Galpha16 cells stably transfected with human hMCH-1R are resuspended using a syringe (needle 0.6x25 mm) and diluted in test buffer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM142203(US8933079, 7.12 | US8933079, 7.13)
Affinity DataIC50:  35nMpH: 7.0Assay Description:Membranes from CHO/Galpha16 cells stably transfected with human hMCH-1R are resuspended using a syringe (needle 0.6x25 mm) and diluted in test buffer...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM142203(US8933079, 7.12 | US8933079, 7.13)
Affinity DataIC50:  67nMpH: 7.0Assay Description:Membranes from CHO/Galpha16 cells stably transfected with human hMCH-1R are resuspended using a syringe (needle 0.6x25 mm) and diluted in test buffer...More data for this Ligand-Target Pair
In DepthDetails US Patent