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Found 2 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50188823'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188823(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human MCH1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50188823(3-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-y...)
Affinity DataIC50:  7.80nMAssay Description:Activity at human MCH1R by GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed