TargetMelanocortin receptor 5(Homo sapiens (Human))
H. Lee Moffitt Cancer Center & Research Institute
Curated by ChEMBL
H. Lee Moffitt Cancer Center & Research Institute
Curated by ChEMBL
Affinity DataKi: 9.90nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:In vitro activaction of mouse recombinant Melanocortin-5 receptor.More data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:Activity in mouse melanocortin-5 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:Agonist activity towards mouse Melanocortin-5 receptor (mMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 0.0710nMAssay Description:Effective concentration against mouse Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.260nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0780nMAssay Description:In vitro agonist potency for Mouse Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0620nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.280nMAssay Description:Agonist activity at mouse MC5 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.170nMAssay Description:Agonistic activity against mouse MC5RMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0780nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0860nMAssay Description:Functional activity at the mouse melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0950nMAssay Description:Effective concentration for mouse Melanocortin-5 receptorMore data for this Ligand-Target Pair