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Found 2 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1A' and Ligand = 'BDBM50464409'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464409(CHEMBL4283539)
Affinity DataKi:  1nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cell membranes after 120 mins by filter binding methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50464409(CHEMBL4283539)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed