Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Ligand = 'BDBM50278288'
Affinity DataKi: 3nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Medical Research Council Technology
Curated by ChEMBL
Medical Research Council Technology
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at mGluR1More data for this Ligand-Target Pair