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Found 3 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 2' and Ligand = 'BDBM212933'
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM212933(US9278960, 4-1 | US9663506, Example 4-1)
Affinity DataIC50:  68nMAssay Description:Negative allosteric modulation of human mGluR2 by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM212933(US9278960, 4-1 | US9663506, Example 4-1)
Affinity DataIC50:  163nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM212933(US9278960, 4-1 | US9663506, Example 4-1)
Affinity DataIC50:  163nMAssay Description:The utility of the compounds in accordance with the present invention as antagonists of metabotropic glutamate receptor activity, in particular mGluR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent