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Found 2 Enz. Inhib. hit(s) with Target = 'Methylated-DNA--protein-cysteine methyltransferase' and Ligand = 'BDBM50068780'
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50068780(6-(Pyridin-4-ylmethoxy)-6,9-dihydro-1H-purin-2-yla...)
Affinity DataIC50:  130nMAssay Description:O6-Alkylguanine-DNA Alkyltransferase-Inactivating Activity (Concentration of inactivator required to produce 50% reduction in ATPase activity) More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethylated-DNA--protein-cysteine methyltransferase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50068780(6-(Pyridin-4-ylmethoxy)-6,9-dihydro-1H-purin-2-yla...)
Affinity DataIC50:  200nMAssay Description:O6-Alkylguanine-DNA Alkyltransferase-Inactivating Activity in Raji cells (Concentration of inactivator required to produce 50% reduction in ATPase ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed